354. S. D. Wood, W. Grant, I. Adrados, J. Y. Choi, J. M. Alburger, D. R. Duckett, W. R. Roush, 'In Silica HTS and Structure Based Optimization of Indazole-Derived ULK1 Inhibitors' ACS Med. Chem. Lett. 2017, 8, 1258. 10.1021/acsmedchemlett.7b00344

353. C. M. Calvet, J. Y. Choi, D. Thomas, B. Suzuki, K. Hirata, S. Lostracco-Johnson, L. B. de Mesquita, A. Nogueira, M. Meuser-Batista, T. A. Silva, J. L. Siqueira-Neto, W. R. Roush, M. C. D. Pereira, J. H. McKerrow, L. M. Podust, '4-aminopyridyl-based lead compounds targeting CYP51 prevent spontaneous parasite relapse in a chronic model and improve cardiac pathology in an acute model of Trypanosoma cruzi infection' PLOS Neglected Tropical Diseases 2017, 11, e0006132. 10.1371/journal.pntd.0006132

352. E. A. Rondini, L. Mladenovic-Ljiljana, W. R. Roush, G. T. Halvorsen, A. E. Green, J. G. Granneman, 'Novel Pharmacological Probes Reveal ABHD5 as a Locus of Lipolysis Control in White and Brown Adipocytess' Journal of Pharmacology and Experimental Therapeutics 2017, 363, 367. 10.1124/jpet.117.243253

351. A.R. Nanna, X. L. Li, E. Walseng, L. Pedzisa, R. S. Goydel, D. Hymel, T. R. Burke, W. R. Roush, C. Rader, 'Harnessing a catalytic lysine residue for the one-step preparation of homogeneous antibody-drug conjugates' Nature Comm. 2017, 8, 2041. 10.1038/s41467-017-01257-1

350. J. Y. Choi, R. Fuerst, A. M. Knapinska, A. B. Taylor, L. Smith, X. H. Cao, P. J. Hart, G. R. Fields, W. R. Roush, 'Structure-Based Design and Synthesis of Potent and Selective Matrix Metalloproteinase 13 Inhibit'ors' J. Med. Chem. 2017, 60, 5816. 10.1021/acs.jmedchem.7b00514

349. C. Allais, W. R. Roush, 'Enantio- and Diastereoselective Synthesis of 1,5-syn-(Z)-Amino Alcohols via Imine Double Allylboration: Synthesis of trans-1,2,3,6-Tetrahydropyridines and Total Synthesis of Andrachcine' Org Lett. 2017, 19, 2649. 10.1021/acs.orglett.7b00995

348. J. W. Mason, C. L. Schmid, L. M. Bohn, W. R. Roush, 'Stolonidiol: Synthesis, Target Identification, and Mechanism for Choline Acetyltransferase Activation' JACS, 2017,139, 5865. 10.1021/jacs.7b01083

347. I. V. Getun, Z. Wu, M. Fallahi, S. Ouizem, Q. Liu, W. Li, R. Costi, W. R. Roush, J. L. Cleveland, P. R. J. Bois, 'Functional Roles of Acetylated Histone Marks at Mouse Meiotic Recombination Hotspots' Mol and Cell Biol. 2017, 37, e00942. 10.1128/MCB.00942-15

346. J. Y. Choi, W. R. Roush, 'Structure Based Design of CYP51 Inhibitors' Current Topics in Med. Chem. 2017, 17, 30. 10.2174/1568026616666160719164933

345. E. Walseng, C. G. Nelson, J. Qi, A. R. Nanna, W. R. Roush, R. K. Goswami, S.C. Sinha, T. R. Burke Jr, C. Rader, 'Chemically Programmed Bispecific Antibodies in Diabody Format' J. Biol. Chem. 2016, 37, 291. 10.1074/jbc.M116.745588

344. J.T. Patterson, H.D. Wilson, S. Asano, N. Nilchan, R.P. Fuller, W.R. Roush, C. Rader, C.F. Barbas, 'Human Serum Albumin Domain I Fusion Protein for Antibody Conjugation' Bioconj. Chem. 2016, 27, 2271. 10.1021/acs.bioconjchem.6b00432

343. L. Pedzisa, X. Li, C. Rader, W.R. Roush, 'Assessment of reagents for selenocysteine conjugation and the stability of selenocysteine adducts' Org. Biomol. Chem. 2016, 14, 5141. 10.1039/C6OB00775A

342. R.N. Nair, J.K. Mishram F.Z. Li, M. Tortosa, C.Y. Yang, J.R. Doherty, M. Cameron, J.L. Cleveland, W.R. Roush, T.D. Bannister, 'Exploiting the co-reliance of tumours upon transport of amino acids and lactate: Gln and Tyr conjugates of MCT1 inhibitors' MedChemComm 2016, 7, 900. 10.1039/c5md00579e

341. B.D. Jones, A. Tochowicz, Y. Tang, M.D. Cameron, L. McCall, K. Hirata, J. L. Siqueirna-Neto, S.L. Reed, J. H. McKerrow, W. R. Roush, "Synthesis and Evaluation of Oxyguanidine Analogues of the Cysteine Protease Inhibitor WRR-483 against Cruzain" ACS Med. Chem. Lett. 2016, 7, 77. 10.1021/acsmedchemlett.5b00336

340. L. H. Rosenberg, M. Lafitte, V. Quereda, W. Grant, W. Chen, M. Bibian, Y. Noguchi, M. Fallahi, C. Yang, J. C. Chang, W. R. Roush, J. L. Cleveland, D. R. Duckett, "Therapeutic targeting of casein kinase 1δ in breast cancer" Science Translational Medicine 2015, 7, 318RA202. 10.1126/scitranslmed.aac8773

339. M. A. Sanders, F. Madoux, L. Mladenovic, H. M. Zhang, X. Q. Ye, M. Angrish, E. P. Mottillo, J. A. Caruso, G. Halvorsen, W. R. Roush, P. Chase, P. Hodder, J. G. Granneman, "Endogenous and Synthetic ABHD5 Ligands Regulate ABHD5-Perilipin Interactions and Lipolysis in Fat and Muscle" Cell Metabolism 2015, 22, 851. doi:10.1016/j.cmet.2015.08.023

338. X. L. Li, J. T. Patterson, M. Sarkar, L. Pedzisa, T. Kodadek, W. R. Roush, C. Rader, "Site-Specific Dual Antibody Conjugation via Engineered Cysteine and Selenocysteine Residues" Bioconjugate Chem. 2015, 26, 2243. 10.1021/acs.bioconjchem.5b00244

337. X. El Hilali, W. R. Roush, "Enantio- and diastereoselective synthesis of syn-beta-hydroxy-alpha-alkenyl carboxamides via reductive aldol reactions of morpholine 4-methyl-2,3-pentadienoic carboxamide with diisopinocampheylborane" Tett. Lett. 2015, 23, 3281. 10.1016/j.tetlet.2015.01.018

336. S. L. Schreiber, J. D. Kotz, M. Li, J. Aubé, C. P. Austin, J. C. Reed, H. Rosen, E. L. White, L. A. Sklar, C. W. Lindsley, B. R. Alexander, J. A. Bittker, P. A. Clemons, A. de Souza, M. A. Foley, M. Palmer, A. F. Shamji1, M. J. Wawer, O. McManus, M. Wu, B. Zou, H. Yu, J. E. Golden, F. J. Schoenen, A. Simeonov, A. Jadhav, M. R. Jackson, A. B. Pinkerton, T. D.Y. Chung, P. R. Griffin, B. F. Cravatt, P. S. Hodder, W. R. Roush, E. Roberts, D. H. Chung, C. B. Jonsson, J. W. Noah, W. E. Severson, S. Ananthan, B. Edwards, T. I. Oprea, P. J. Conn, C. R. Hopkins, M. R. Wood, S. R. Stauffer, and K. A. Emmitte 'Advancing Biological Understanding and Therapeutics Discovery with Small-Molecule Probes' Cell. 2015, 6, 1252. 10.1016/j.cell.2015.05.023

335. C. Penas, E. Govek, Y. Fang, V. Ramachandran, M. Daniel, W. Wang, M. Maloof, R. Rahaim, M. Bibian, D. Kawauchi, D. Finkelstein, J. Han, J. Long, B. Li, D. Robbins, M. Malumbres, M. Roussel, W. Roush, M. Hatten, N. Ayad, "Casein Kinase 1 delta Is an APC/C-Cdh1 Substrate that Regulates Cerebellar Granule Cell Neurogenesis," Cell Rep. 2015, 11, 249. 10.1016/j.celrep.2015.03.016

334. L. McCall, A. Aroussi, J. Choi, D. Vieira, G. De Muylder, J. Johnson, S. Chen, D. Kellar, J. Siqueira-Neto, W. Roush, L. Podust, J. McKerrow, "Targeting Ergosterol Biosynthesis in Leishmania donovani: Essentiality of Sterol 14alpha-demethylase," PLOS Neglected Tropical Diseases. 2015, 9, 1. 10.1371/journal.pntd.0003588

333. H. Ghalei, F. X. Schaub, J. R. Doherty, Y. Noguchi, W. R. Roush, J. L. Cleveland, M. E. Stroupe, and K. Karbstein, “CK1d-directed release of Ltv1 from pre-40S ribosomes is necessary for risobome assembly and cellular growth,” J. Cell Biol. 2015, 6, 745. 10.1083/jcb.201409056

332. Y. Wang, R. L. Stowe, C. E. Pinello, G. Tian, F. Madoux, D. Li, L. Y. Zhao, J.-L. Li, K. R. Geary, H. Ma, P. Hodder, W. R. Roush, and D. Liao, “Identification of novel small-molecule HDAC inhibitors that selectively inhibit class I HDACs and kill cancer cells through HDAC inhibition,” Chemistry & Biology, 2014, 22, 273. 10.1016/j.chembiol.2014.12.015

331. C. Corzo, Y. Mari, M. R. Chang, D. Kuruvilla, P. Nuhant, N. Kumar, G. M. West, D. Duckett, W. R. Roush, and P. R. Griffin, “Anti-proliferation activity of a small molecule repressor of LRH1,” Mol. Pharmacol. 2014, in press.  

330. D. F. Vieira, J. Y. Choi, C. M. Calvet, J. L. Siqueira-Neto, J. B. Johnston, D. Kellar, J. Gut, M. D. Cameron, J. H. McKerrow, W. R. Roush and L. M. Podust, “Binding mode and potency of N-indolyl-oxopyridinyl-4-aminopropanyl-based inhibitors targeting Trypanosoma cruzi CYP51,” J. Med. Chem. 2014, 57,10162. 10.1021/jm501568b

329. T. P. Spicer, J. Jiang, A. B. Taylor, P. J. Hart, W. R. Roush, G. B. Fields, Peter S. Hodder, and D. Minond, “Characterization of Selective Exosite-Binding Inhibitors of Matrix Metalloproteinase 13 That Prevent Articular Cartilage Degradation In Vitro”, J. Med. Chem. 2014, 57, 9598. 10.1021/jm501284e

328. C. Penas, J. K. Mishra, S. D. Wood, S. C. Schurer, W. R. Roush and N. G. Ayad, “GSK3 Inhibitors Stabilize Wee1 and Reduce Cerebellar Granule Cell Progenitor Proliferation,” Cell Cycle, 2015, 14, 417. 10.4161/15384101.2014.974439

327. J. Y. Choi, L. Podust, and W. R. Roush, “Drug Strategies Targeting CYP51 in Neglected Tropical Diseases,” Chem. Rev. 2014, 114, 11242. 10.1021/cr5003134

326. C.M Calvet, D.F. Vieira, J.Y. Choi, D. Kellar, M.D. Cameron, J.L. Siqueira-Neto, J. Gut, J.B. Johnson, L. Lin, S. Khan, J.H. McKerrow, W.R. Roush, L.M. Podust, "4-Aminopyridyl-Based CYP51 Inhibitors as Anti-Trypanosoma cruzi Drug Leads with Improved Pharmacokinetic Profile and in Vivo Potency," J. Med. Chem. 2014, 6989-7005. 10.1021/jm500448u

325. H. Wang, C. Yang, J. R. Doherty, W. R. Roush, J. L. Cleveland, T. D. Bannister, “Synthesis and Structure Activity Relationships of Pteridine Dione and Trione Monocarboxylate Transporter 1 Inhibitors,” J. Med. Chem. 2014, 57, 7317. 10.1021/jm500640x

324. C. Penas, V. Ramachandran, S. Simanski, C. Lee, F. Madoux, R. J. Rahaim, R. Chauhan, O. Barnaby, S. Schurer, P. Hodder, J. Steen, W. R. Roush, and N. G. Ayad, “Casein Kinase 1d Dependent Wee1 Degradation,” J. Biol. Chem. 2014, 289, 18893. 10.1074/jbc.M114.547661

323. D. F. Vieira, J. Y. Choi, W. R. Roush,] and L. M. Podust, "Expanding the Binding Envelope of CYP51 Inhibitors Targeting Trypanosoma cruzi with 4-Aminopyridyl-Based Sulfonamide Derivatives," ChemBioChem, 2014, 1111. 10.1002/cbic.201402027

322. J. Y. Choi, C. M. Calvet, D. F. Vieira, S. S. Gunatilleke, M. D. Cameron, J. H. McKerrow, L. M. Podust, and W. R. Roush, "R-Configuration of 4-Aminopyridyl-Based Inhibitors of CYP51 Confers Superior Efficacy Against Trypanosoma cruzi," Med. Chem. Lett. 2014, 434. 10.1021/ml500010m

321. J. R. Doherty, C. Yang, K. E. N. Scott, M. D. Cameron, M. Fallahi, W. Li, M. A. Hall, A. L. Amelio, J. K. Mishra, F. Li, M. Tortosa, H. M. Genau, R. J. Rounbehler, Y. Lu, C. V. Dang, K. G. Kumar, A. A. Butler, T. D. Bannister, A. Hooper, K. Unsal-Kacmaz, W. R. Roush and J. L. Cleveland, “Blocking lactate export by inhibiting the Myc target Mct1 Disables Glycolysis and Glutathione Metabolism,” Cancer Res. 201474, 908-920. 10.1158/0008-5472.CAN-13-2034

320. J. Kister, D. S. Ess, and W. R. Roush, "Enantio- and Diastereoselective Synthesis of syn-β-Hydroxy-α-Vinyl Carboxylic Esters via Reductive Aldol Reactions of Ethyl Allenecarboxylate with 10-TMS-9-Borabicyclo[3.3.2]decane and DFT Analysis of the Hydroboration Pathway,"Org. Lett. 2013, 15, 5436. 10.1021/ol4025277

C. Allais, A. S. Tsai, P. Nuhant, and W. R. Roush, "Highly Diastereo- and Enantioselective Aldol Reactions of Stereodefined Tetrasubstituted Enolborinates Generated By 1,4- Hydroboration of α,β-Unsaturated Morpholine Carboxamides with
(Diisopinocampheyl)borane," Angew. Chem. Int. Ed. 2013, 52, 12888–12891. 10.1002/anie.201307302

J. Y. Choi, C. M. Calvet, S. S. Gunatilleke, C. Ruiz, M. D. Cameron, J. H. McKerrow, L. M. Podust, and W. R. Roush, "Rational development of 4-aminopyridyl-based inhibitors targeting 22 Trypanosoma cruzi CYP51 as anti-Chagas agents," J. Med. Chem., 2013, 56, 7651. 10.1021/jm401067s

C. Allais, P. Nuhant, and W. R. Roush, "(Diisopinocampheyl)borane-Mediated ReductiveAldol Reactions of Acrylate Esters: Enantioselective Synthesis of Anti-Aldols," Org. Lett. 2013, 15, 3922. 10.1021/ol401679g

M. Chen and W. R. Roush, "Enantioselective Synthesis of (Z)-2-Methyl-1,5-anti- and (E)-2- Methyl-1,5-anti-Pentenediols Via an Allene Hydroboration-Double Allylboration Reaction Sequence," J. Am. Chem. Soc. 2013, 135, 9512. 10.1021/ja4033633

P. Nuhant, C. Allais and W. R. Roush, "(Diisopinocampheyl)borane-Mediated Reductive Aldol Reactions: Highly Enantio- and Diastereoselective Synthesis of Syn-Aldols from NAcryloylmorpholine," Angew. Chem. Int. Ed. 2013, 52, 8703.

M. Bibian, R. J. Rahaim, J. Y. Choi, Y. Noguchi, S. Schürer, W. Chen, S. Nakanishi, K. Licht, L. H. Rosenberg, L. Li, Y. Feng, M. D. Cameron, D. R. Duckett, J. L. Cleveland and W. R. Roush, "Development of Highly Selective Casein Kinase 1δ/1ε (CK1δ/ε) Inhibitors with Potent Antiproliferatve Properties," Bioorg. Med. Chem. Lett. 2013, 23, 4374. 10.1016/j.bmcl.2013.05.075

M. Chen and W. R. Roush, "Enantiodivergent Hydroboration Reactions of a Racemic Allenylsilane with Diisopinocampheyl-borane and Curtin-Hammett Controlled Double Asymmetric Crotylboration Reactions of (S)-E-α-Phenyldimethylsilyl-
(ddiisopinocampheyl)crotylborane," Tetrahedron 2013, 69, 5468 and 7551. (Invitedmanuscript for Tetrahedron Symposium-in-Print in honor of Prof. Paul Wender's 2013 Tetrahedron Prize). 10.1016/j.tet.2013.06.053

P. Nuhant and W. R. Roush, "Enantio- and Diastereoselective Synthesis of N-Acetyl Dihydrotetrafibricin Methyl Ester," J. Am. Chem. Soc. 2013, 135, 5340. 10.1021/ja401918r

M. Chen and W. R. Roush, "Enantioselective Synthesis of (E)-δ-Silyl-anti Homoallylic Alcohols Via An Enantiodivergent Hydroboration-Crotylboration Reaction of a Racemic Allenylsilane", Org. Lett., 2013, 15 1622. 10.1021/ol4004405

H. Yang, C. Pinello, J. Luo, D. Li, Y. Wang, L. Zhao, S. Jahn, A. Saldanha, B. Law, W. Roush, P. Hodder, and D. Liao, "Small-molecule inhibitors of acetyltransferase p300 identified by high-throughput screening are potent anticancer agents", Mol. Cancer Therap. 2013, in press.

A. S. Tsai, M. Chen and W. R. Roush, "Chiral Bronsted Acid Catalyzed Enantioselective Synthesis of anti-Homopropargyl Alcohols via Kinetic Resolution-Aldehyde Allenylboration Using Racemic Allenylboronates," Org. Lett. 2013, 15, in press. 10.1021/ol4003459

J. R. Abbott and W. R. Roush, "Stereoselective Synthesis of the Disaccharide Unit of Incednine," Org. Lett. 2013, 15, 62. 10.1021/ol303093z

J. G. Geist, R. Barth and W. R. Roush, "Enantioselective Synthesis of the C(1) - C(11) Fragment of Tedanolide C", Org. Lett. 2013, 15, 58. 10.1021/ol303089w

M. Chen and W. R. Roush, “Crotylboron-Based Synthesis of the Polypropionate Units of Chaxamycins A/D, Salinisporamycin, and Rifamycin S,” J. Org. Chem. 2012, 77, in press. 10.1021/jo3008226

305.  J.-L. Han, M. Chen and W. R. Roush, “Diastereo- and Enantioselective Synthesis of (E)-2-Methyl-1,2-anti-3- pentanediols via Allenylboronate Kinetic Resolution with (dIpc)2BH and Aldehyde Allylboration,” Org. Lett. 2012, 14, 3028. 10.1021/ol3010968

304. M. Chen and W. R. Roush, “Enantioselective Synthesis of anti- and syn-Homopropargyl Alcohols via Chiral Brønsted Acid Catalyzed Asymmetric Allenyboration Reactions,” J. Am. Chem. Soc. 2012, 134, 1094710947. 10.1021/ja3031467

303. A. T. Dossey, J. Whitaker, M. C. A. Dancel, R. Vander Meer, U. R. Bernier, M. Gottardo, and W. R. Roush, “Defensive Spiroketals from Asceles glaber (Phasmatodea): Absolute Configuration and Effects on Ants and Mosquitoes,J. Chem. Ecol. 2012, 38, 1105.

302.  M. Chen and W. R. Roush, “Enantioselective Synthesis of  (+)-Crocacin C.  An Example of A Highly Challenging Mismatched Double Asymmetric d-Stannylcrotylboration Reaction,” Org. Lett., 2012, 14, 1880.10.1021/ol300476f

301. M. Chen and W. R. Roush, “Enantioselective Synthesis of (-)-Basiliskamide A,” Org. Lett., 2012, 14, in press (ASAP). 10.1021/ol300282e

300.  M. Chen and W. R. Roush, “Highly Stereoselective Synthesis of Anti, Anti-Steriotriads:  A Solution to the Challenging Mismatched Double Asymmetric Crotylboration Reactions,” J. Am. Chem. Soc., 2012, 134, 3925. 10.1021/ja300472a

299.  J. Y. Choi, M. S. Plummer, J. Starr, C. R. Desbonnet, H. Soutter, J. Chang, J. R. Miller, K. Dillman, A. A. Miller, and W. R. Roush, "Structure Guided Development of Novel Thymidine Mimetics Targeting Pseudomonas aeruginosa Thymidylate Kinase: From Hit to Lead Generation,” J. Med. Chem. 2012, 55, 852-870. 10.1021/jm201349f

298.  M. Chen and W. R. Roush, “Total Synthesis of (-)-Tirandamycin C,” Org. Lett. 2012, 14, 426. 10.1021/ol203161u

297.  M. Ying and W. R. Roush, “"Studies on the Synthesis of Reidispongiolide A:  Stereoselective Synthesis of the C(22)-C(36) Fragment,” Tetrahedron 2011, 67, 10274 (invited paper for Symposium-in-Print in honor of Prof. G. Stork’s 90th birthday). 10.1016/j.tet.2011.10.029

296.  J. Roth, D. Minond, E. Darout, Q. Liu, J. Lauer, P. Hodder, G. B. Fields, and W. R. Roush, “Identification of Novel, Exosite-Binding Matrix Metalloproteinase-13 Inhibitor Scaffolds,” Bioorg. Med. Chem. Lett. 2011, 21, 7180-7184. 10.1016/j.bmcl.2011.09.077

295.  Y. Zhou, J. Agudelo, K. Lu, D. H. Goetz, E. Hansell, Y. T. Chen, W. R. Roush, J. McKerrow, C. S. Craik, S. M. Amberg, and G. Simmons, “Inhibitors of SARS-CoV Entry - Identification using an Internally-Controlled Dual Envelope Pseudovirion Assay,” Antiviral Res2011, 92, 187-194. 10.1016/j.antiviral.2011.07.016

294.  H. Sun, J. R. Abbott, and W. R. Roush, “Stereoselective Synthesis of a Model C(18)-C(35) Spiroketal Fragment of Integramycin,” Org. Lett201113, 2734. 10.1021/ol200834p

293.  P. Nuhant, J. Kister, R. Lira, A. Sorg and W. R. Roush, “Development of a Double Allylboration Reagent Targeting 1,5-syn-(E)-Diols:  Application to the Synthesis of the C(23)-C(40) Fragment of Tetrafibricin,” Tetrahedron 201167, 6497. (invited paper for Symposium-in-Print in honor of Prof. S. Omura's Tetrahedron Prize). Corrigendum: 2012, 68, 774.10.1016/j.tet.2011.06.008

 L.A. Solt, N. Kumar, P. Nuhant, Y. Wang, J. L. Lauer, J. Liu, M. Istrate, T. M. Kamenecka, W. R. Roush, D. Vidovic, S. C. Schurer, J. Xu, G. Wagoner, P. D. Drew, P. R. Griffin and T. P. Burris, "Inhibition of the TH17 Differentiation and Suppression of Autoimmunity by a Selective Synthetic ROR Ligand," Nature 2011, 472, 491. 10.1038/nature10075

 M. Chen and W. R. Roush, “Enantioselective Syntheses of syn- and antiI- β-Hydroxyallylsilanes via Allene Hydroboration-Aldehyde Allylboration Reactions,” Org. Lett. 2011, 13, 1992. 10.1021/ol200392u

 M. Chen and W. R. Roush, “Enantioconvergent Hydroboration of a Racemic Allene: Enantioselective Synthesis of (E)-d- Stannyl-anti-Homoallylic Alcohols via Aldehyde Crotylboration,” J. Am. Chem. Soc. 2011, 133, 5744. 10.1021/ja2010187

289.  J. Kister, P. Nuhant, R. Lira, A. Sorg and W. R. Roush, “Enantio- and Diastereoselective Syntheses of (E)-1,5-syn-Diols:  Application to the Synthesis of the C(23)-C(40) Fragment of Tetrafibricin,”Org. Lett. 2011, 13 , 1868. 10.1021/ol2003836

288.  S. A. Busby, N. Kumar, D. S. Kuruvilla, M. A. Istrate, J. J. Conkright, Y. Wang, T. M. Kamenecka, M. D. Cameron, W. R. Roush, T. P. Burris and P. R. Griffin, “Identification of a Novel Non-retinoid Pan Inverse Agonist of the Retinoic Acid Receptors,” ACS Chem. Biol. 2011, ASAP. 10.1021/cb100396s

287.  Y. Lee, J. Y. Choi, H.  Fu, C. Harvey, S. Ravindran, W. Roush, J. C. Boothroyd, and C. Khosla, “Chemistry and Biology of Macrolide Antiparasitic Agents,” J. Med. Chem., 2011, 54, 2792. 10.1021/jm101593u

286.  P. Stewart, M. Chen, W. R. Roush, and D. Ess, “Thermodynamic Control of 1,3-Boratropic Shifts of α- and γ-Stannyl-Substituted Allylboranes:  Hyperconjugation Outweighs Steric Effects,” Org. Lett. 2011, 13, 1478. 10.1021/ol2001599

285.  N. Kumar, D. J. Kojetin, L. A. Solt, K. G. Kumar, P. Nuhant, D. R. Duckett, M. D. Cameron, A. A. Butler, W. R. Roush, P. R. Griffin and T. P. Burris, “Identification of SR3335 (ML176), a Synthetic RORa Selective Inverse Agonist,” ACS Chem. Biol. 2011, 6, 218. 10.1021/cb1002762

284.  H. Sun and W. R. Roush, “Synthesis of (S,S)-Diisopropyl Tartrate (E)-Crotylboronate and Its Reaction with Aldehydes: (2R,3R,4R)-1,2-Dideoxy-2-ethenyl-4,5-O-(1-methylethylidene)-xylitol,” Org. Synth. 2011, 88, 181.

283.  H. Sun and W. R. Roush, “Synthesis of (+)-B-Allyldiisopinocampheylborane and Its Reaction with Aldehydes: (2R, 3R)-1-(tert-Butyldiphenylsilyloxy)-2-methylhex-5-en-3-ol,” Org. Synth. 2011, 88, 87.

282.  J. T. Halvorsen and W. R. Roush, “Stereoselective Synthesis of the Decahydrofluorene Core of the Hirsutellones,” Tetrahedron Lett. 2011, in press (invited manuscript for special issue in honor of Prof. Harry Wasserman’s 90th birthday). 10.1016/j.tetlet.2010.10.111