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Scientific Report 2008
Chemistry
Chairman's Overview
Staff
K.C. Nicolaou, Ph.D.*
Chairman
Aline W. and L.S. Skaggs Professor of
Chemical Biology
Darlene Shiley Chair in Chemistry
Dariush Ajami, Ph.D.
Assistant Professor of Molecular Assembly
Phil S. Baran, Ph.D.
Professor
Dale L. Boger, Ph.D.*
Richard and Alice Cramer Professor of
Chemistry
Tobin J. Dickerson, Ph.D.
Assistant Professor
Sheng Ding, Ph.D.
Associate Professor
Albert Eschenmoser, Ph.D.*
Professor
M.G. Finn, Ph.D.*
Professor
Valery Fokin, Ph.D.
Associate Professor
M. Reza Ghadiri, Ph.D.*
Professor
William A. Greenberg, Ph.D.
Assistant Professor of Chemistry
Inkyu Hwang, Ph.D.
Assistant Professor
Kim D. Janda, Ph.D.**
Professor
Ely R. Callaway, Jr., Chair in
Chemistry
Director, Worm Institute of Research
and Medicine
Gunnar Kaufmann, Ph.D.
Assistant Professor of Chemistry
Jeffery W. Kelly, Ph.D.*
Lita Annenberg Hazen Professor of Chemistry
Ramanarayanan Krishnamurthy, Ph.D.
Associate Professor
Lucas J. Leman, Ph.D.
Assistant Professor of Chemistry
Richard A. Lerner, M.D.***
President, The Scripps Research Institute
Lita Annenberg HazenProfessor of
Immunochemistry
Cecil H. and Ida M. Green Chair in Chemistry
Roy Periana, Ph.D.*****
Professor
Evan T. Powers, Ph.D.
Associate Professor of Chemistry
Julius Rebek, Jr., Ph.D.*
Professor
Director, The Skaggs Institute for Chemical
Biology
Edward Roberts, Ph.D.
Professor
Floyd E. Romesberg, Ph.D.
Associate Professor
William Roush, Ph.D.*****
Professor
Peter G. Schultz, Ph.D.*
Professor
Scripps Family Chair
K. Barry Sharpless, Ph.D.*
W.M. Keck Professor of Chemistry
Anita D. Wentworth, Ph.D.
Assistant Professor
Paul Wentworth, Jr., Ph.D.
Professor
Chi-Huey Wong, Ph.D.*
Professor of Chemistry
Jin-Quan Yu, Ph.D.
Associate Professor
(Andrew) Bin Zhou, Ph.D.
Assistant Professor of Immunochemistry
SENIOR SCIENTIST
Luis Martinez, Ph.D.*****
Staff Scientists
Lisa Eubanks, Ph.D.
Rajesh Grover, Ph.D.
Sarah Hanson, Ph.D.
Lubica Supekova, Ph.D.
Wen Xiong, Ph.D.
Instrumentation/service Facilities
Raj K. Chadha, Ph.D.
Director, X-ray Crystallography Facility
Dee H. Huang, Ph.D.
Director, Nuclear Magnetic Resonance
Facility
Gary E. Siuzdak, Ph.D.
Senior Director, Mass Spectrometry Facility
Senior Research Associate
Suresh Pitram, Ph.D.
Research Associates
Ramzey Abujarour, Ph.D.
Rajesh Ambasudhan, Ph.D.
Manuel Amorin Lopez, Ph.D.
Mark Ams, Ph.D.
Yoshio Ando, Ph.D.
Deepshikha Angrish, Ph.D.
Shinji Ashida, Ph.D.
Micahel Baksh, Ph.D.
Deboshri Banerjee, Ph.D.
Elizabeth Barrett, Ph.D.****
Roland Barth, Ph.D.*****
Clay Bennett, Ph.D.
Moritz Biskup, Ph.D.
Universität Karlsruhe
Karlsruhe, Germany
Anthony Boitano, Ph.D.
Genomics Institute of the Novartis Foundation
San Diego, California
Laure Bouchez, Ph.D.
Kristopher Boyle, Ph.D.
Christopher Burke, Ph.D
Antonio Burtoloso, Ph.D.
University of Sao Paulo
Sao Paulo, Brazil
Mark Bushey, Ph.D.
Exxon, Inc.
Union City, New Jersey
Darren Bykowski, Ph.D.*****
Petr Capek, Ph.D.
Katerina Capkova, Ph.D.
Arani Chanda, Ph.D.
Ke Chen, Ph.D.
Peng Chen, Ph.D.
Govardhan Cherukupalli, Ph.D.
Epix Pharmaceuticals
Lexington, Massachusetts
Jodie Chin, Ph.D.
Srinivas Reddy Chirapu, Ph.D.
Chandramouli Chiruta, Ph.D.
Dong-Gyu Cho, Ph.D.
So-Hye Cho, Ph.D.
Sungwook Choi, Ph.D.
Joyanta Choudhury, Ph.D.
Sarwat Chowdhury, Ph.D.
Stepan Chuprakov, Ph.D.
Petr Cigler, Ph.D.
T. Ryan Cirz
Achaogen
South San Francisco, California
Scott Cockroft, Ph.D.
University of Edinburgh
Edinburgh, Scotland
David Colby, Ph.D.
Purdue University
West Lafayette, Indiana
Kevin Cole, Ph.D.
Eli Lilly and Company
Indianapolis, Indiana
Christine Crane, Ph.D.
Matthew Cremeens, Ph.D.
Gonzaga University
Redmond, Washington
Fernando Rodrigo Pinacho Crisostomo,
Ph.D.
Burnham Institute for Medical Research
La Jolla, California
Jeffrey Culhane, Ph.D.
Stephen Dalby, Ph.D.
Etzer Darout, Ph.D.
Pfizer Inc.
Groton, Connecticut
Amy DeBaillie, Ph.D.
Eli Lilly and Company
Indianapolis, Indiana
Judith Denery, Ph.D.
Ross Denton, Ph.D.
University of Cambridge
Cambridge, England
Caroline Desponts, Ph.D.
Antonia Di Mola, Ph.D.
Deguo Du, Ph.D.
Anna Dubrovska, Ph.D.
Viktoriya Dubrovskaya, Ph.D.
Joshua Dunetz, Ph.D.
Pfizer Inc.
Groton, Connecticut
Kyle Eastman, Ph.D.
David Edmonds, Ph.D.
Jem Efe, Ph.D.
Jan Elsner, Ph.D.
Celgene Pharmaceuticals
San Diego, California
Daniel Ess, Ph.D.
Cyrine Ezzili, Ph.D.
Xingang Fang, Ph.D.
Simon Ficht, Ph.D.
Sanofi-Aventis Deutschland GmbH
Frankfurt, Germany
Joseph Rodolph Fotsing, Ph.D.
Senomyx, Inc.
San Diego, California
Bozena Frackowiak, Ph.D.
Politechnika Opolska
Opole, Poland
Graeme Freestone, Ph.D.
Metabasis Therapeutics, Inc.
San Diego, California
Yu Fu, Ph.D.
Amelia Fuller, Ph.D.
Santa Clara University
Santa Clara, California
Jianmin Gao, Ph.D.
Boston College
Chestnut Hill, Massachusetts
Haibo Ge, Ph.D.
Savvas Georgiades, Ph.D.****
Ola Ghoneim, Ph.D.
Qatar University
Doha, Qatar
Nathan Gianneschi, Ph.D.
University of California
San Diego, California
Cristina Gil-Lamaignere, Ph.D.
University Hospital Nuestra Señora
de la Candelaria
Santa Cruz de Tenerife, Spain
Rodolfo Gonzalez, Ph.D.
Scott Grecian, Ph.D.
Neil Grimster, Ph.D.
Rajesh K. Grover, Ph.D.
Jan Grunewald, Ph.D.
Tanja Gulder, Ph.D.
Richard Guy, Ph.D.****
Masaki Handa, Ph.D.
Sagami Chemical Research Center
Ayase, Kanagawa, Japan
Yuanjun He, Ph.D.
Jason Hein, Ph.D.
Dube Henry, Ph.D.
Marcos Hernandez, Ph.D.
Par Holmberg, Ph.D.
Memorial Sloan Kettering Cancer Center
New York, New York
Wen-Xu Hong, Ph.D.
Zhangyong Hong, Ph.D.
Richard J. Hooley, Ph.D.
University of California
Riverside, California
Tamara Hopkins, Ph.D.
Boehringer Ingelheim Pharmaceuticals,
Inc.
Ridgefield, Connecticut
Allen Horhota, Ph.D.
Tony Horneff, Ph.D.
Jun-Li Hou, Ph.D.
Claas Hovelmann, Ph.D.
Fang Hu, Ph.D.
Department of Molecular Biology, Scripps
Research
Xiaoyi Hu, Ph.D.
Zheng-Zheng Huang, Ph.D.
DuPont Central Research and Development
Wilmington, Delaware
Ben Hutchins, Ph.D.
Der-ren Hwang, Ph.D.
Academia Sinica
Taipei, Taiwan
Giltae Hwang, Ph.D.
Michael Jahnz, Ph.D.
NOXXON Pharma AG
Berlin, Germany
Rong Jiang, Ph.D.*****
Guo Jiantoa, Ph.D.
Hiroyuki Kakei, Ph.D.
Takeda Pharmaceutical Company Limited
Osaka, Japan
Jaroslaw Kalisiak, Ph.D.
Seiji Kamioka, Ph.D.
Moumita Kar, Ph.D.
Kwang Mi Kim, Ph.D.
F. Scott Kimball, Ph.D.
Jeremy Kister, Ph.D.
Keith Korthals, Ph.D.
Larisa Krasnova, Ph.D.
Arkady Krasovskiy, Ph.D.
Luke Lairson, Ph.D.
Jae Wook Lee, Ph.D.
Jinq-Chyi Lee, Ph.D.
National Health Research Institutes
Miaoli County, Taiwan
Jong Seok Lee, Ph.D.
Ki-Bum Lee, Ph.D.
Rutgers University
Piscataway, New Jersey
Sejin Lee, Ph.D.
SK Drug Development Center
Daejong, Korea
Alexandre Lemire, Ph.D.****
Edward Lemke, Ph.D.
Christophe Letondor, Ph.D.****
Chuang-Chuang Li, Ph.D.
Peking University
Peking, China
Fangzheng Li, Ph.D.*****
Hongming Li, Ph.D.
Schering-Plough
Kenilworth, New Jersey
Ke Li, Ph.D.
DuPont Central Research and Development
Wilmington, Delaware
Pi-Hui Liang, Ph.D.
Academia Sinica
Taipei, Taiwan
Yeon-Hee Lim, Ph.D.
Schering-Plough
Kenilworth, New Jersey
Tongxiang Lin, Ph.D.
Troy Lister, Ph.D.
Novartis
Cambridge, Massachusetts
Christopher Liu, Ph.D.
Cubix Pharmaceuticals
Lexington, Massachusetts
Wenshe Liu, Ph.D.
Texas A&M University
College Station, Texas
Michael Luzung, Ph.D.
Utpal Majumder, Ph.D.
Sreeman Mamidyala, Ph.D.
Takeshi Masuda, Ph.D.
Michael Maue, Ph.D.
Bayer CropScience AG
Monheim, Germany
Alexander Mayorov, Ph.D.
Charles Melancon, Ph.D.
Lionel Moisan, Ph.D.
CEA
Gif-Sur-Yvette, France
Ana Montero, Ph.D.****
Miguel Morales, Ph.D.
Adam Morgan, Ph.D.
Concert Pharmaceuticals, Inc.
Lexington, Massachusetts
Ting-Wei Mu, Ph.D.
S. Vasudeva Naidu, Ph.D.
Yuya Nakai, Ph.D.
Joonwoo Nam, Ph.D.
CytRx Corporation
San Diego, California
Tae-Gyu Nam, Ph.D.
Andrew Nguyen, M.D., Ph.D.
Romain Noel, Ph.D.
George Nora, Ph.D.*****
Severin Odermatt, Ph.D.****
Christian Olsen, Ph.D.
Yazmin Osornio, Ph.D.****
Junguk Park, Ph.D.
Nitin Patil, Ph.D.
Johan Paulsson, Ph.D.
Richard Payne, Ph.D.
University of Sydney
Sydney, Australia
Xuemei Peng, Ph.D.****
Murali Peram Surakattula, Ph.D.
CytRx Corporation
San Diego, California
Roshan Perera, Ph.D.
University of Texas
Austin, Texas
Ramulu Poddutoori, Ph.D.
Jonathan Pokorski, Ph.D.
Agustì Lledó Ponsati, Ph.D.
Daniela Radu, Ph.D.
DuPont Central Research and Development
Wilmington, Delaware
Ronald Rahaim, Ph.D.*****
Praveen Rao, Ph.D.
University of Waterloo
Waterloo, Ontario, Canada
Per Restorp, Ph.D.
Kimberly Reynolds, Ph.D.
Jin-Kyu Rhee, Ph.D.
Fatima Rivas, Ph.D.
Joshua Roth, Ph.D.*****
Troy Ryba, Ph.D.
Broad Institute of MIT and Harvard
Cambridge, Massachusetts
Youngha Ryu, Ph.D.
Texas Christian University
Fort Worth, Texas
Catherine Saccavini, Ph.D.
Nicholas Salzameda, Ph.D.
Antonio Sanchez-Ruiz, Ph.D.
Yoshikazu Sasaki, Ph.D.
Stefan Schiller, Ph.D.
Niklas Schone, Ph.D.
Michael Schramm, Ph.D.
California State University
Long Beach, California
Young Jun Seo, Ph.D.
Edward Sessions, Jr., Ph.D.
Shigeki Seto, Ph.D.
Mary Jo Sever, Ph.D.
Alex Shaginian, Ph.D.
Ardea Biosciences
San Diego, California
David Shaw, Ph.D.
Weijun Shen, Ph.D.
Xiao Shengxiong, Ph.D.
Bingfeng Shi, Ph.D.
Yan Shi, Ph.D.
Hiroki Shigehisa, Ph.D.
Hiroyuki Shimamura, Ph.D.
Siddhartha Shenoy, Ph.D.
Ryan Simkovsky, Ph.D.
Chinnappan Sivasankar, Ph.D.****
Michael Smolinski, Ph.D.
Kinex Pharmaceuticals
Buffalo, New York
Xinyi Song, Ph.D.
Simon Stamm, Ph.D.
Sebastian Steiniger, Ph.D.
Antonia Stepan, Ph.D.
James Stover, Ph.D.
Bernhard Stump, Ph.D.
Shun Su, Ph.D.
Hui Kai Sun, Ph.D.*****
Shinobu Takizawa, Ph.D.
Adam Talbot, Ph.D.
Institute of Chemical and Engineering
Sciences
Jurong Island, Singapore
Annie Tam, Ph.D.
Yefeng Tang, Ph.D.
Mariola Tortosa, Ph.D.
Instituto de Quimica Organica, CSIC
Madrid, Spain
Craig Turner, Ph.D.****
Matthew Tremblay, Ph.D.
Vincent Trepanier, Ph.D.
Institute of Chemical and Engineering
Sciences
Jurong Island, Singapore
Jonathan Tripp, Ph.D.
Meng-Lin Tsao, Ph.D.
University of California
Merced, California
Andrew Udit, Ph.D.
Taiki Umezawa, Ph.D.
Hokkaido University
Sapporo, Japan
Kenji Usui, Ph.D.
Tokyo Institute of Technology
Tokyo, Japan
Carlos Valdez, Ph.D.
Rigel Pharmaceuticals, Inc.
South San Francisco, California
Punna Venkateshwarlu, Ph.D.
Feng Wang, Ph.D.
Jian Wang, Ph.D.
Jiangyun
Wang, Ph.D.
Institute of Biophysics
Beijing, China
Lin Wang, Ph.D.
Sheng-Kai Wang, Ph.D.
Weidong Wang, Ph.D.
Xisheng Wang, Ph.D.
Yajuan Wang, Ph.D.
Yuanhua Wang, Ph.D.
Timo Weide, Ph.D.
Albert Willis, Ph.D.
Pharmagra Labs, Inc.
Brevard, North Carolina
Tao Wu, Ph.D.
Institute of Chemical and Engineering
Sciences
Jurong Island, Singapore
Heiko Wurdak, Ph.D.
Jian Xie, Ph.D.
Wen Xiong, Ph.D.
Yue Xu, Ph.D.
Junichiro Yamaguchi, Ph.D.
Ryu Yamasaki, Ph.D.
Tokyo University of Science
Tokyo, Japan
Ura Yasuyuki, Ph.D.
Nara Women's University
Nara, Japan
Yan Yin, Ph.D.
Ian Young, Ph.D.
Zhanqian Yu, Ph.D.
Xu Yuan, Ph.D.
Weiqiang Zhan, Ph.D.
Hongjun Zhang, Ph.D.
Xuejun Zhang, Ph.D.
Yanghui Zhang, Ph.D.
Yingchao Zhang, Ph.D.
Hoffmann-La Roche, Inc.
Nutley, New Jersey
Heyue Zhou, Ph.D.
Hongyan Zhou, Ph.D.
Shoutian Zhu, Ph.D.
Joerg Zimmermann, Ph.D.
Visiting Investigators
Keisuke Fukuchi, Ph.D.
Sankyo Co., Ltd.
Tokyo, Japan
Christine Hernandez, Ph.D.
University of Philippines
Diliman, Philippines
(Edmond) Shie-Liang Hsieh, Ph.D.
National Yang-Ming University
Taipei, Taiwan
Masakazu Imamura, Ph.D.
Astellas Pharma Inc.
Tsukuba, Ibaraki, Japan
Kuniyuki Kishikawa, Ph.D.
Kyowa Hakko Kogyo Co., Ltd.
Sunto-gun, Shizuoka, Japan
Michael Meijler, Ph.D.
Ben-Gurion University of the Negev
Be'er Sheva, Israel
Takayoshi Suzuki, Ph.D.
Nagoya City University
Nagoya, Japan
Yoshiyuki Yoneda, Ph.D.
Daiichi Pharmaceutical Co., Ltd.
Tokyo, Japan
Scientific Associate
Jon Ashley
* Joint appointment in The Skaggs Institute for Chemical Biology
** Joint appointments in The
Skaggs Institute for Chemical Biology and the Department of Immunology and Microbial
Science
*** Joint appointments in The Skaggs Institute for Chemical Biology and the Department of Molecular Biology
**** Appointment completed
***** Scripps Florida
Appointment completed; new location shown
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