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Authors, Title Journal, Volume, Pages, (Year) |
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Willis, B., Eubanks, L.M., Wood, M.R., Janda, K.D., Dickerson, T.J., Lerner, R.A.L., "Biologically templated organic polymers with nanoscale order" PNAS, 105(5), 1416 (2008) |
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Brogan, A.P., Dickerson, T.J., Janda, K.D., "Nornicotine-organocatalyzed aqueous reduction of alpha, beta-unsaturated aldehydes" Chem. Commun., 46, 4952 (2007) |
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Capcova, K., Yoneda, Y., Dickerson, T.J., Janda, K.D., "Synthesis and structure-activity relationships of second-generation hydroxymate botulinum neurotoxin A protease inhibitors" Bioorg. Med. Chem. Lett., 17, 6463 (2007) |
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Xu, Y., Hixon, M.S., Dawson, P.E., Janda, K.D., "Development of o FRET assay for monitoring of HIV gp41 core disruption" J. Org. Chem., 72(18), 6700 (2007) |
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McAllister, L.A., Hixon, M.S., Schwartz, R., Kubitz, D.S., Janda, K.D., "Synthesis and application of a novel ligand for affinity chromatography based removal of endotoxin from antibodies" Bioconj. Chem., 18, 559 (2007) |
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Brogan, A.P., Dickerson, T.J., Janda, K.D., "Enamine-based aldol organocatalysis in water: Are they really "all wet"?" Angew. Chem. Int. Ed., 45, 8100 (2006) |
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Xu, Y., Lu, H., Kennedy, J.P., Yan, X., McAllister, L.A., Yamamoto, N., Moss, J.A., Boldt, G.E., Jiang, S., Janda, K.D., "Evaluation of "credit-card" libraries for inhibition of HIV-1 gp41 fusogenic core formation" J. Comb. Chem., 8, 531 (2006) |
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Xu, Y., Shi, J., Yamamoto, N., Moss, J.A., Vogt, P.K., Janda, K.D., "A credit-card library approach for disrupting protein-protein interactions" Bioorg. Med. Chem., 14, 2660 (2006) |
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Moss, J.A., Stokols, S., Hixon, M.S., Ashley, F.T., Chang, J.Y., Janda, K.D., "Solid-phase synthesis and kinetic characterization of fluorogenic enzyme-degradable hydrogel cross-linkers" Biomacromolecules, 7, 1011 (2006) |
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Boldt, G.E., Dickerson, T.J., Janda, K.D., "Emerging chemical and biological approaches for the preparation of discovery libraries" Drug Disc. Today, 11, 143 (2006) |
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Rogers, C.J., Dickerson, T.J., Janda, K.D., "Kinetic isotope and thermodynamic analysis of the nornicotine-catalyzed aqueous aldol reaction" Tetrahedron, 62, 352 (2006) |
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Shimomura, O., Lee, B.S., Meth, S., Suzuki, H., Mahajan, S., Nomura, R., Janda, K.D., "Synthesis and application of polytetrahydrofuran-grafted polystyrene (PS-PTHF) resin supports for organic synthesis" Tetrahedron, 61, 12160 (2005) |
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Rogers, C.J., Dickerson, T.J., Wentworth, Jr.,P., Janda, K.D., "A high-swelling reagent scaffold suitable for use in aqueous and organic solvents" Tetrahedron, 61, 12140 (2005) |
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Zhang, L., Long, H., Boldt, G.E., Janda, K.D., Schatz, G.C., Lewis, F.D., "alpha- and beta-Stilbenosides as base-pair surrogates in DNA hairpins" Org. Biomol. Chem., 4, 314 (2006) |
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Qi, L., Yamamoto, N., Meijler, M.M., Altobell, III, L.J., Koob, G.F., Wirsching, P., Janda, K.D., "Delta-9-tetrahydrocannabinol immunochemical studies: Haptens, monoclonal antibodies, and a convenient synthesis of radiolabeled delta-9-tetrahydrocannabinol" J. Med. Chem., 48, 7389 (2005) |
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Shute, T.S., Matsushita, M., Dickerson, T.J., La Clair, J.J., Janda, K.D., Burkart, M.D., "A site-specific bifunctional protein labeling system for affinity and fluorescent analysis" Bioconjugate Chem., 16, 1352 (2005) |
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Yamashita, M., Lee, S.-H., Koch, G., Zimmermann, J., Clapham, B., Janda, K.D., "Solid-phase synthesis of oxazolones and other heterocycles via Wang resin-bound diazocarbonyls" Tetrahedron Lett., 46, 5495 (2005) |
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Lee, B.S., Mahajan, S., Janda, K.D., "Molecular iodine-catalyzed imine activation for three-component nucleophilic addition reactions" Synlett, 8, 1325 (2005) |
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Lee,B.S., Mahajan, S., Janda, K.D., "Asymmetric dihydroxylation catalyzed by ionic polymer-supported osmium tetroxide" Tetrahedron Lett., 46, 4491 (2005) |
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Rogers, C.L., Dickerson, T.J., Brogan, A.P., Janda,K.D., "Hammett correlation of nornicotine analogues in the aqueous aldol reaction: Implications for green organocatalysis" J. Org. Chem., 70(9), 3705 (2005) |
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Lee, B.S., Mahajan, S., Janda, K.D., "Cross-linked poly(4-vinylpyridine/styrene) copolymers as a support for immobilization of ytterbium triflate" Tetrahedron, 61, 3081 (2005) |
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Reed, N.N., Dickerson, T.J., Boldt, G.E., Janda, K.D., "Enantioreversal in the Sharpless asymmetric epoxidation reaction controlled by the molecular weight of a covalently appended achiral polymer" J. Org. Chem., 70(5), 1728 (2005) |
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Lee, B.S., Mahajan, S., Janda, K.D., "Novel method for catalyst immobilization using an ionic polymer: A case study using recyclable yttterbium triflate" Tetrahedron Letters, 46, 807 (2005) |
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Lee, S.-H., Yoshida, K., Matsushita, H., Clapham, B., Koch, G., Zimmermann, J., Janda, K.D., "N-H insertion reactions of primary ureas: The synthesis of highly substituted imidazolones and imidazoles from diazocarbonyls" J. Org. Chem., 69, 8829 (2004) |
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Matsushita, H., Lee, S.-H., Yoshida, K., Clapham, B., Koch, G., Zimmermann, J., Janda, K.D., "N-H insertion reactions of Boc-amino acid amides: Solution- and solid-phase synthesis of pyrazinones and pyrazines" Org. Lett., 6, 4627 (2004) |
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Lee, B.-S., Mahajan, S., Clapham, B., Janda, K.D., "Suspension ring-opening metathesis polymerization: The preparation of norbornene-based resins for application in organic synthesis" J. Org. Chem., 69, 3319 (2004) |
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Lee, S.-H., Matsushita, H., Clapham, B., Janda, K.D., "The direct conversion of carbamates to ureas using aluminum amides" Tetrahedron, 60, 3439 (2004) |
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Matsushita, H., Lee, S.-H., Joung, M., Clapham, B., Janda, K.D., "Smart cleavage reactions: the synthesis of benzimidazoles and benzothiazoles from polymer-bound esters" Tetrahedron Letters, 45, 313 (2004) |
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Chen, Y., Gambs, C., Abe, Y., Wentworth, P., Jr., Janda, K.D., " Total synthesis of the depsipeptide FR-901375" J.Org. Chem., 68, 8902 (2003) |
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Dickerson, T.J., Reed, N.N., Janda, K.D., "Soluble polymers as catalyst and reagent platforms: Liquid-phase methodologies" In: Polymeric Materials in Organic Synthesis and Catalysis ed. M.R. Buchmeiser, Wiley-VCH Verlag Gmbh, Weinheim, Germany, pp 241-276 (2003) |
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Shimomura, O., Clapham, B., Spanka, C., Mahajan, S., Janda, K.D., "Application of microgels as polymer supports for organic synthesis: Preparation of a small phthalide library, a scavenger, and a borohydride reagent" J. Comb. Chem., 4, 436 (2002) |
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Delgado, M., Janda, K.D., "Polymeric supports for solid phase organic synthesis" Current Organic Chemistry, 6, 1031 (2002) |
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Kim, G.-T., Wenz, M., Park, J.-I., Hasserodt, J., Janda, K.D., "Polyene substrates with unusual methylation patterns to probe the active sites of three catalytic antibodies" Biorg. Med. Chem., 10, 1249 (2002) |
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Isomura, S., Hoffman, T.Z., Wirsching, P., Janda, K.D., "Synthesis, properties, and reactivity of cocaine benzoylthio ester possessing the cocaine absolute configuration" J. Amer. Chem. Soc., 124, 3661 (2002) |
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Cordova, A., Tremblay, M.R., Clapham, B., Janda, K.D., "A sequential application of kinetic resolution and polymer-supported scavenging for the isolation of chiral secondary alcohols" J. Org. Chem., 66, 5645 (2001) |
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Lee, K.J., Janda, K.D., "Traceless solid-phase synthesis of 5-Benzoylbenzimidazoles" Can. J. Chem., 79, 1556 (2001) |
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Clapham, B., Reger, T.S., Janda, K.D., "Polymer-supported catalysis in synthetic organic chemistry" Tetrahedron, 57, 4637 (2001) |
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Brummer, O., Clapham, B., Janda, K.D., "Solid-phase synthesis of oligoesters using a JandaJel resin" Tetrahedron Letters, 42, 2257 (2001) |
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Wen, K., Han, H., Hoffman, T.Z., Janda, K.D., Orgel, L.E., "The synthesis of Beta-peptides containing guanidino groups" Bioorg. Med. Chem. Lett., 11, 689 (2001) |
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Cordova, A., Janda, K.D., "A highly chemo- and stereoselective synthesis of Beta-keto esters via a polymer-supported lipase catalyzed transesterification" J. Org. Chem., 66, 1906 (2001) |
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Clapham, B., Cho, C.-W., Janda, K.D., "A polymer-supported proline-based diamine catalyst for the kinetic resolution of racemic secondary alcohols" J. Org. Chem., 66, 868 (2001) |
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Manzotti, R., Reger, T.S., Janda, K.D., "Improved synthesis of (4-ethenylphenyl)diphenyl methanol and its application in the preparation of trityl functionalized polystyrene resin containing tetrahydrofuran derived cross-linker" Tetrahedron Letters, 41, 8417 (2000) |
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Tremblay, M.R., Wentworth, P. Jr., Lee, G.E. Jr., Janda, K.D., "Parallel solid-phase synthesis and structural characterization of a library of highly substituted chiral 1,3-oxazolidines" J. Comb. Chem., 2, 698 (2000) |
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Sieber, F., Wentworth, P. Jr., Janda, K.D., "Exploiting poly(ethylene glycol) as a matrix for liquid-phase organic synthesis" Molecules, 5, 1018 (2000) |
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Manzotti, R., Tang, S.-Y., Janda, K.D., "Improved synthesis of prostanoids on a non-cross-linked polystyrene soluble support" Tetrahedron, 56, 7885 (2000) |
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Vaino, A.R., Janda, K.D., "Solid phase organic synthesis: A critical understanding of the resin" J. Comb. Chem., 2, 579 (2000) |
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Reed, N.N., Janda, K.D., "A one step synthesis of monoprotected polyethylene glycol ethers" J. Org. Chem., 65, 5843 (2000) |
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Hasserodt, J., Janda, K.D., Lerner, R.A., "A class of 4-aza-lithocholic acid-derived haptens for the generation of catalytic antibodies with steroid synthase capabilities" Bioorg. Med. Chem., 8, 995 (2000) |
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Harwig, C.W., Hoffman, T.Z., Wentworth, A.D., Janda, K.D., "A one-pot multistep approach to alpha-azido-phospohonate and phosphonothioate diesters: Key intermediates in the synthesis of haptens for the generation of antibody ligases" Bioorg. Med. Chem. Lett., 10, 915 (2000) |
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Toy, P.H., Reger, T.S., Janda, K.D., "Soluble polymer bound cleavage reagents: A multipolymer strategy for the cleavage of tertiary amines from REM resin" Org. Lett., 2, 2205 (2000) |
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Brummer, O., Clapham, B., Janda, K.D., "Recent developments and applications of polymer-supported reagents in synthetic organic chemistry" Current Opinion in Drug Discovery & Dev., 3, 462 (2000) |
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Toy, P.H., Janda, K.D., "Soluble polymer-supported organic synthesis" Acc. Chem. Res., 33, 546 (2000) |
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Reger, T.S., Janda, K.D., "Polymer-supported (Salen)Mn catalysts for asymmetric epoxidation: A comparison between soluble and insoluble matrices" J. Am. Chem. Soc., 122, 6929 (2000) |
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Lopez-Pelegrin, J.A., Janda, K.D., "Solution- and soluble-polymer supported asymmetric syntheses of six-membered ring prostanoids" Chem. Eur. J., 6, 1917 (2000) |
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Wentworth, A.D., Wentworth, P. Jr., Mansoor, F.U., Janda, K.D., "A soluble polymer-supported triflating reagent: A high-throughput synthetic approach to aryl and enol triflates" Org. Lett., 2, 477 (2000) |
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Lee, K.J., Angulo, A., Ghazal, P., Janda, K.D., "Soluble-polymer supported synthesis of a prostanoid library: Identification of antiviral activity" Org. Lett., 1, 1859 (1999) |
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Wentworth, P. Jr., Janda, K.D., "Liquid-phase chemistry: Recent advances in soluble polymer-supported catalysts, reagents and synthesis" Chem. Commun., 1917 (1999) |
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Cordova, A., Reed, N.N., Ashley, J.A., Janda, K.D., "Convenient synthesis of L-proline benzyl ester" Bioorg. Med. Chem. Lett., 9, 3119 (1999) |
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Brummer, O., Wentworth, P. Jr., Weiner, D.P., Janda, K.D., "Phosphorodithioates: Synthesis and evaluation of new haptens for the generation of antibody acyl transferases" Tetrahedron Letters, 40, 7307 (1999) |
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Han, H., Cho, C.-W., Janda, K.D., "A substrate-based methodology that allows the regioselective control of the catalytic aminohydroxylation reaction" Chem. Eur. J., 5, 1565 (1999) |
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Berg, T., Simeonov, A., Janda, K.D., "A combined parallel synthesis and screening of macrocyclic lanthanide complexes for the cleavage of phospho di- and triesters and double-stranded DNA" J. Comb. Chem., 1, 96 (1999) |
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Yoon, J., Cho, C.-W., Han, H., Janda, K.D., "Solution and soluble polymer synthesis of 3-aminoimidazoline-2,4-diones" Chem. Commun., 2703 (1998) |
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Chen, S., Janda, K.D., "Total synthesis of naturally occurring prostaglandin F2-alpha on a non-cross-linked polystyrene support" Tetrahedron Letters, 39, 3943 (1998) |
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Yli-Kauhaluoma, J.T., Harwig, C.W., Wentworth, P. Jr., Janda, K.D., "Unexpected 1,3-oxazolidine formation in the attempted oxidation of N-aryl-N-methyl substituted Beta-amino alcohols using pyridinium dichromate" Tetrahedron Letters, 39, 2269 (1998) |
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Han, H., Yoon, J., Janda, K.D., "An efficient asymmetric route to 2,3-diaminobutanoic acids" J. Org. Chem., 63, 2045 (1998) |
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Gravert, D.J., Janda, K.D., "Bifunctional initiators for free radical polymerization of non-crosslinked block copolymers" Tetrahedron Letters, 39, 1513 (1998) |
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Hori, M., Janda, K.D., "A soluble polymer approach to the "Fishing Out" principle: Synthesis and purification of Beta-Amino alcohols" J. Org. Chem., 63, 889 (1998) |
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Gravert, D.J., Janda, K.D., "Synthesis on soluble polymers: New reactions and the construction of small molecules" Current Opinion in Chemical Biology, 1, 107 (1997) |
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Chen, S., Janda, K.D., "Synthesis of prostaglandin E2 methyl ester on a soluble-polymer support for the construction of prostanoid libraries" J. Am. Chem. Soc., 119, 8724 (1997) |
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Hasserodt, J., Janda, K.D., "Syntheses of octahydroquinoline-N-oxides: Haptens designed to elicit catalytic antibodies that control a terpenoid-like cascade cyclization" Tetrahedron, 53, 11237 (1997) |
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Han, H., Janda, K.D., "Multipolymer-supported substrate and ligand approach to the Sharpless asymmetric dihydroxylation," Angew. Chem. Int. Ed., 36, 1731 (1997) |
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Wentworth, P. Jr., Janda, K.D., "Synthesis of oxorhenium (V) and oxotechnetium (V) complexes as inhibitors of ribonucleases and for the generation of catalytic antibodies" Synlett, 5, 537 (1997) |
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Han, H., Janda, K.D., "A soluble polymer-bound approach to the Sharpless catalytic asymmetric dihydroxylation (AD) reaction: Preparation and application of a [(DHQD)2 PHAL-PEG-OMe] ligand" Tetrahedron Letters, 38, 1527 (1997) |
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Wentworth, P. Jr., Wiemann, T., Janda, K.D., "A new class of pentacoordinate ribonuclease inhibitors: Synthesis, characterization and inhibition studies of ribonucleoside and anhydropentofuranose oxorhenium (V) complexes" J. Am. Chem. Soc., 118, 12521 (1996) |
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Wentworth, P. Jr., Janda, K.D., "A facile and efficient route to 3',5'-diamino-3',5'-dideoxynucleosides" Chem. Commun., 2097 (1996) |
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Sakurai, M., Wirsching, P., Janda, K.D., "Design and synthesis of a cocaine-diamide hapten for vaccine development" Tetrahedron Letters, 37, 5479 (1996) |
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Han, H., Yoon, J., Janda, K.D., "Azatides: Solution and Liquid phase Syntheses" In: Peptidomimetics, Methods in Molecular Biology series, Humana Press, Inc., eds. W.M. Kazmierski, (1996) |
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Jung, K.W., Sanfilippo, P.J., Wachter, M., Janda, K.D., "Syntheses and biological evaluation of two new naproxen analogs" Bioorg. Med. Chem. Lett., 6, 2281 (1996) |
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Han, H., Janda, K.D., "Soluble polymer-bound ligand-accelerated catalysis: Asymmetric dihydroxylation" J. Am. Chem. Soc., 118, 7632 (1996) |
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Sakurai, M., Wirsching, P., Janda, K.D., "Synthesis of a nucleoside hapten with a [P(O)-O-N] linkage to elicit catalytic antibodies with phosphodiesterase activity" Bioorg. Med. Chem. Lett., 6, 1055 (1996) |
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Lavey, B.J., Janda, K.D., "Applying Antibody Catalysis to Organic Synthesis" In: Antibody Expression and Engineering, ACS Symposium Series 604, eds., H.Y. Wang, T. Imanaka, Chapter 10, p.123 (1995) |
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Fenniri, H., Janda, K.D., Lerner, R.A., "Encoded reaction cassette for the highly sensitive detection of the making and breaking of chemical bonds" Proc. Natl. Acad. Sci. USA, 92, 2278 (1995) |
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Yli-Kauhaluoma, J., Janda, K.D., "An expedient synthesis of isopropyl anisoles and veratroles" Tetrahedron Letters, 35, 4509 (1994) |
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