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Authors, Title
Journal, Volume, Pages, (Year) |
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Boldt, G.E., Dickerson, T.J., Janda, K.D., "Emerging chemical and biological approaches for the preparation of discovery libraries"
Drug Disc. Today, 11, 143 (2006) |
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Shimomura, O., Lee, B.S., Meth, S., Suzuki, H., Mahajan, S., Nomura, R., Janda, K.D., "Synthesis and application of polytetrahydrofuran-grafted polystyrene (PS-PTHF) resin supports for organic synthesis"
Tetrahedron, 61, 12160 (2005) |
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Rogers, C.J., Dickerson, T.J., Wentworth, Jr.,P., Janda, K.D., "A high-swelling reagent scaffold suitable for use in aqueous and organic solvents"
Tetrahedron, 61, 12140 (2005) |
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Dickerson, T.J., Beuscher IV, A.E., Rogers, C.J., Hixon, M.S., Yamamoto, N., Xu, Y., Olson, A.J., Janda, K.D. , "Discovery of acetylcholinesterase peripheral anionic site ligands through computational refinement of a directed library"
Biochemistry, 44, 14845 (2005) |
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Lee, B.S., Mahajan, S., Janda, K.D., "Cross-linked poly(4-vinylpyridine/styrene) copolymers as a support for immobilization of ytterbium triflate"
Tetrahedron, 61, 3081 (2005) |
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Reed, N.N., Dickerson, T.J., Boldt, G.E., Janda, K.D., "Enantioreversal in the Sharpless asymmetric epoxidation reaction controlled by the molecular weight of a covalently appended achiral polymer"
J. Org. Chem., 70(5), 1728 (2005) |
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Lee, B.S., Mahajan, S., Janda, K.D., "Novel method for catalyst immobilization using an ionic polymer: A case study using recyclable yttterbium triflate"
Tetrahedron Letters, 46, 807 (2005) |
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Lee, S.-H., Yoshida, K., Matsushita, H., Clapham, B., Koch, G., Zimmermann, J., Janda, K.D., "N-H insertion reactions of primary ureas: The synthesis of highly substituted imidazolones and imidazoles from diazocarbonyls"
J. Org. Chem., 69, 8829 (2004) |
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Matsushita, H., Lee, S.-H., Yoshida, K., Clapham, B., Koch, G., Zimmermann, J., Janda, K.D., "N-H insertion reactions of Boc-amino acid amides: Solution- and solid-phase synthesis of pyrazinones and pyrazines"
Org. Lett., 6, 4627 (2004) |
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Lee, S.-H., Matsushita, H., Koch, G., Zimmermann, J., Clapham, B., Janda, K.D., "Smart cleavage reactions: the synthesis of an array of ureas from polymer-bound carbamates"
J. Comb. Chem., 6, 822 (2004) |
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Lee, B.-S., Mahajan, S., Clapham, B., Janda, K.D., "Suspension ring-opening metathesis polymerization: The preparation of norbornene-based resins for application in organic synthesis"
J. Org. Chem., 69, 3319 (2004) |
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Matsushita, H., Lee, S.-H., Joung, M., Clapham, B., Janda, K.D., "Smart cleavage reactions: the synthesis of benzimidazoles and benzothiazoles from polymer-bound esters"
Tetrahedron Letters, 45, 313 (2004) |
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Lee, S.-H., Clapham, B., Koch, G., Zimmerman, J., Janda, K.D., "Solid-phase rhodium carbenoid N-H insertion reactions: the synthesis of a diverse array of indoles"
J. Comb. Chem., 5, 188 (2003) |
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Fujimori, T., Wirsching, P., Janda, K.D., "Preparation of a Krohnke pyridine combinatorial library suitable for solution-phase biological screening"
J. Comb. Chem., 5, 625 (2003) |
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Dickerson, T.J., Reed, N.N., Janda, K.D., "Soluble polymers as catalyst and reagent platforms: Liquid-phase methodologies"
In: Polymeric Materials in Organic Synthesis and Catalysis ed. M.R. Buchmeiser, Wiley-VCH Verlag Gmbh, Weinheim, Germany, pp 241-276 (2003) |
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Gambs, C., Dickerson, T.J., Mahajan, S., Pasternack, L.B., Janda, K.D., "High-resolution diffusion-ordered spectroscopy to probe the microenvironment of JandaJel and Merrifield resins"
J. Org. Chem., 68(9), 3673 (2003) |
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Ahn, J.-A., Wentworth, Jr., P., Janda, K.D., "Soluble polymer-supported convergent parallel library synthesis"
Chem. Commun., 480 (2003) |
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Lee, S.-H., Clapham, C., Koch, G., Zimmermann, J., Janda, K.D., "Rhodium carbenoid N-H insertion reactions of primary ureas: Solution and solid-phase synthesis of imidazolones"
Org. Lett., 5(4), 511 (2003) |
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Dickerson, T.J., Reed, N.N., Janda, K.D., "Soluble polymers as scaffolds for recoverable catalysts and reagents"
Chem. Rev., 102, 3325 (2002) |
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Shimomura, O., Clapham, B., Spanka, C., Mahajan, S., Janda, K.D., "Application of microgels as polymer supports for organic synthesis: Preparation of a small phthalide library, a scavenger, and a borohydride reagent"
J. Comb. Chem., 4, 436 (2002) |
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Clapham, B., Lee, S.-H., Koch, G., Zimmermann, J., Janda, K.D., "The preparation of polymer bound Beta-ketoesters and their conversion into an array of oxazoles"
Tetrahedron Letters, 43, 5407 (2002) |
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Ahn, J.-M., Boyle, N.A., MacDonald, M.T., Janda, K.D., "Peptidomimetics and peptide backbone modifications"
Mini Reviews in Medicinal Chemistry, 2, 463 (2002) |
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Delgado, M., Janda, K.D., "Polymeric supports for solid phase organic synthesis"
Current Organic Chemistry, 6, 1031 (2002) |
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Reed, N.N., Delgado, M., Hereford, K., Clapham, B., Janda, K.D., "Preparation of soluble and insoluble polymer supported IBX reagents"
Bioorg. Med. Chem. Lett., 12, 2047 (2002) |
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Janda, K.D., "(Preface) Polymer supported catalysts and reagents in synthetic organic chemistry, Bioorg."
Med. Chem. Lett., 12, vii (2002) |
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Spanka, C. Wentworth, Jr., P., Janda, K.D., "Developing soluble polymers for high-throughput synthetic chemistry"
Combinatorial Chemistry and High Throuput Screening, 5, 233 (2002) |
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Delgado, M., Lee, K.J., Altobell, III, L., Spanka, C., Wentworth, Jr., P., Janda, K.D., "A parallel approach to the discovery of carrier delivery vehicles to enhance antigen immunogenicity"
J. Amer. Chem. Soc., 124, 4946 (2002) |
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Spanka, C., Clapham, B., Janda, K.D., "Preparation of new microgel polymers and their application as supports in organic synthesis"
J. Org. Chem., 67, 3045 (2002) |
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Boyle, N.A., Janda, K.D., "Formats for combinatorial synthesis: solid-phase, liquid-phase and surface"
Current Opinion in Chemical Biology, 6, 339 (2002) |
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Reger, T.S., Janda, K.D., "Parallel suspension polymerization for high-throughput resin synthesis"
Bioorg. Med. Chem., 12, 837 (2002) |
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Delgado, M., Spanka, C., Kerwin, L.D., Wentworth, Jr., P., Janda, K.D., "A tunable hydrogel for encapsulation and controlled release of bioactive proteins"
Biomacromolecules, 3, 262 (2002) |
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Moss, J.A., Dickerson, T.J., Janda, K.D., "Solid phase peptide synthesis on JandaJel resin"
Tetrahedron Letters, 43, 37 (2002) |
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Dickerson, T., Reed, N.N., Janda, K.D., "Regio-reactive resin: A platform for orthogonal loading using the polymer backbone and cross-linker"
Bioorg. Med. Chem. Lett., 11, 1507 (2001) |
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Clapham, B., Reger, T.S., Janda, K.D., "Polymer-supported catalysis in synthetic organic chemistry"
Tetrahedron, 57, 4637 (2001) |
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Brummer, O., Clapham, B., Janda, K.D., "Solid-phase synthesis of oligoesters using a JandaJel resin"
Tetrahedron Letters, 42, 2257 (2001) |
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Toy, P.H., Reger, T.S., Garibay, P., Garno, J.C., Malikayil, J.A., Liu, G.-Y., Janda, K.D., "Polytetrahydrofuran cross-linked polystyrene resins for solid-phase organic synthesis"
J. Comb. Chem., 3, 117 (2001) |
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Toy, P.H., Reger, T.S., Janda, K.D., "Tailoring polystyrene solid-phase synthesis resins: Incorporation of flexible cross-linkers"
Aldrichimica Acta, 33, 87 (2000) |
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Lopez-Pelegrin, J.A., Wentworth, P. Jr., Sieber, F., Metz, W.A., Janda, K.D., "Soluble polymer-supported chemoenzymatic synthesis of the C21-C27 fragment of the Bryostatins"
J. Org. Chem., 65, 8527 (2000) |
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Tremblay, M.R., Wentworth, P. Jr., Lee, G.E. Jr., Janda, K.D., "Parallel solid-phase synthesis and structural characterization of a library of highly substituted chiral 1,3-oxazolidines"
J. Comb. Chem., 2, 698 (2000) |
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Manzotti, R., Tang, S.-Y., Janda, K.D., "Improved synthesis of prostanoids on a non-cross-linked polystyrene soluble support"
Tetrahedron, 56, 7885 (2000) |
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Vaino, A.R., Janda, K.D., "Solid phase organic synthesis: A critical understanding of the resin"
J. Comb. Chem., 2, 579 (2000) |
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Wentworth, P. Jr., Janda, K.D., "A tool-box of polymer matrices for the combinatorial chemist / biotechnologist"
International Convention on Agriculture, Biotechnology and Chemistry; Rome, Italy, p. 211 (2000) |
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Manzotti, R., Janda, K.D., "Solid and liquid phase chemistry: Development of new supports for solid phase organic synthesis and for liquid phase chemistry"
Chimica Oggi/Chemistry Today, 18, 14 (2000) |
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Vaino, A.R., Goodin, D.B., Janda, K.D., "Investigating resins for solid phase organic synthesis: The relationship between swelling and microenvironment as probed by EPR and fluorescence spectroscopy"
J. Comb. Chem., 2, 330 (2000) |
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Vaino, A.R., Janda, K.D., "Euclidean shape-encoded combinatorial chemical libraries"
Proc. Natl. Acad. Sci. USA, 97, 7692 (2000) |
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Toy, P.H., Reger, T.S., Janda, K.D., "Soluble polymer bound cleavage reagents: A multipolymer strategy for the cleavage of tertiary amines from REM resin"
Org. Lett., 2, 2205 (2000) |
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Brummer, O., Clapham, B., Janda, K.D., "Recent developments and applications of polymer-supported reagents in synthetic organic chemistry"
Current Opinion in Drug Discovery & Dev., 3, 462 (2000) |
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Toy, P.H., Janda, K.D., "Soluble polymer-supported organic synthesis"
Acc. Chem. Res., 33, 546 (2000) |
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Reger, T.S., Janda, K.D., "Polymer-supported (Salen)Mn catalysts for asymmetric epoxidation: A comparison between soluble and insoluble matrices"
J. Am. Chem. Soc., 122, 6929 (2000) |
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Lopez-Pelegrin, J.A., Janda, K.D., "Solution- and soluble-polymer supported asymmetric syntheses of six-membered ring prostanoids"
Chem. Eur. J., 6, 1917 (2000) |
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Reed, N.N., Janda, K.D., "Stealth star polymers: A new high-loading scaffold for liquid-phase organic synthesis"
Org. Lett., 2, 1311 (2000) |
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Wentworth, A.D., Wentworth, P. Jr., Mansoor, F.U., Janda, K.D., "A soluble polymer-supported triflating reagent: A high-throughput synthetic approach to aryl and enol triflates"
Org. Lett., 2, 477 (2000) |
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Sieber, F., Wentworth, P. Jr., Janda, K.D., "Exploring the scope of poly(ethylene glycol) (PEG) as a soluble matrix for the Stille cross-coupling reaction"
J. Comb. Chem., 1, 540 (1999) |
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Lee, K.J., Angulo, A., Ghazal, P., Janda, K.D., "Soluble-polymer supported synthesis of a prostanoid library: Identification of antiviral activity"
Org. Lett., 1, 1859 (1999) |
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Wentworth, P. Jr., Janda, K.D., "Liquid-phase chemistry: Recent advances in soluble polymer-supported catalysts, reagents and synthesis"
Chem. Commun., 1917 (1999) |
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Garibay, P., Toy, P.H., Hoeg-Jensen, T., Janda, K.D., "Application of a new solid-phase resin: Benzamide ortho-lithiation and the synthesis of a phthalide library"
Synlett, 9, 1438 (1999) |
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Toy, P.H., Janda, K.D., "New supports for solid-phase organic synthesis: Development of polystyrene resins containing tetrahydrofuran derived cross-linkers"
Tetrahedron Letters, 40,, 6329 (1999) |
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Sieber, F., Wentworth, P. Jr., Toker, J.D., Wentworth, A.D., Metz, W.A., Reed, N.N., Janda, K.D., "Development and application of a poly(ethylene glycol)-supported triarylphosphine reagent: Expanding the sphere of liquid-phase organic synthesis"
J. Org. Chem., 64, 5188 (1999) |
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Han, H., Yoon, J., Janda, K.D., "Azatides as Peptidomimetics / Solution and Liquid Phase Syntheses"
In: Peptidomimetics Protocols, (Methods in Molecular Medicine series), ed. W.M. Kazmierski, Humana Press, Totowa, N.J., Vol. 23, p. 87 (1999) |
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Yoon, J., Han, H., Janda, K.D., "Solution and Soluble Polymer Syntheses of Azatides and Azapeptides"
In: Advances in Amino Acid Mimetics and Peptidomimetics, ed., A. Abell , JAI Press, Inc., Stamford, CT., Vol. 2, p. 247 (1999) |
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Harwig, C.W., Gravert, D.J., Janda, K.D., "Soluble polymers: New options in both traditional and combinatorial synthesis"
Org. Chem. Chemtracts, 12, 1 (1999) |
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Zhao, X.-Y., Janda, K.D., "Soluble polymer traceless linker investigations: Solvent effects on the desulfonylation of polyethylene glycol (PEG) substituted aryl alkyl sulfones with sodium amalgam"
Bioorg. Med. Chem. Lett., 8, 2439 (1998) |
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Yoon, J., Cho, C.-W., Han, H., Janda, K.D., "Solution and soluble polymer synthesis of 3-aminoimidazoline-2,4-diones"
Chem. Commun., 2703 (1998) |
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Zhao, X.-Y., Metz, W.A., Sieber, F., Janda, K.D., "Expanding on the purification methodology of polyethylene glycol (PEG) bound molecules: The synthesis of 3,5-Pyrazolidinediones"
Tetrahedron Letters, 39, 8433 (1998) |
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Hori, M., Gravert, D.J., Wentworth, P. Jr., Janda, K.D., "Investigating highly crosslinked macroporous resins for solid phase synthesis"
Bioorg. Med. Chem. Lett., 8, 2363 (1998) |
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Gravert, D.J., Datta, A., Wentworth, P. Jr., Janda, K.D., "Soluble supports tailored for organic synthesis: Parallel polymer synthesis via sequential normal/living free radical processes"
J. Am. Chem. Soc., 120, 9481 (1998) |
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Berg, T., Vandersteen, A.M., Janda, K.D., "High-throughput synthesis and direct screening for the discovery of novel hydrolytic metal complexes"
Bioorg. Med. Chem. Lett., 8, 1221 (1998) |
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Gravert, D.J., Janda, K.D., "Bifunctional initiators for free radical polymerization of non-crosslinked block copolymers"
Tetrahedron Letters, 39, 1513 (1998) |
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Hori, M., Janda, K.D., "A soluble polymer approach to the "Fishing Out" principle: Synthesis and purification of Beta-Amino alcohols"
J. Org. Chem., 63, 889 (1998) |
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Wentworth, P. Jr., Janda, K.D., "Generating and analyzing combinatorial chemistry libraries"
Current Opinion in Biotechnology, 9, 109 (1998) |
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Gravert, D.J., Janda, K.D., "Synthesis on soluble polymers: New reactions and the construction of small molecules"
Current Opinion in Chemical Biology, 1, 107 (1997) |
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Han, H., Vandersteen, A., Janda, K.D., "Combinatorics, Peptide Mimetics and Combizymes"
In: Peptides: Frontiers of Peptide Science (Proceedings of the 15th American Peptide Symposium) eds., J.P. Tam , T. Pravin, P. Kaumaya, Kluwer/Escom, Nashville, TN., p.22 (1997) |
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Janda, K.D., Gravert, D.J., "Organic reactions on soluble polymer supports as an alternative methodology for combinatorial solid-phase synthesis"
Biotechnology Internl., 169 (1997) |
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Gravert, D.J., Janda, K.D., "Soluble polyethylene glycol supports for liquid-phase combinatorial synthesis"
Drugs of the Future, 22, 1147 (1997) |
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Chen, S., Janda, K.D., "Synthesis of prostaglandin E2 methyl ester on a soluble-polymer support for the construction of prostanoid libraries"
J. Am. Chem. Soc., 119, 8724 (1997) |
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Han, H., Janda, K.D., "Multipolymer-supported substrate and ligand approach to the Sharpless asymmetric dihydroxylation,"
Angew. Chem. Int. Ed., 36, 1731 (1997) |
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Zhao, X.-Y., Janda, K.D., "Syntheses of alkylated malonates on a traceless linker derived soluble polymer support"
Tetrahedron Letters, 38, 5437 (1997) |
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Gravert, D.J., Janda, K.D., "Organic synthesis on soluble polymer supports: Liquid-phase methodologies"
Chemical Reviews, 97, 489 (1997) |
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Jung, K.W., Zhao, X.-Y., Janda, K.D., "Development of new linkers for the formation of aliphatic C-H bonds on polymeric supports"
Tetrahedron, 53, 6645 (1997) |
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Wentworth, P. Jr., Vandersteen, A.M., Janda, K.D., "Poly(ethylene glycol) (PEG) as a reagent support: The preparation and utility of PEG-triarylphosphine conjugate in liquid-phase organic synthesis (LPOS)"
Chem. Commun., 759 (1997) |
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Janda, K.D., A Book Review on, "Combinatorial Peptide and Nonpeptide Libraries : A Handbook by G. Jung, pub: VCH (1996)"
J. Amer. Chem. Soc., 119, 3848 (1997) |
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Han, H., Janda, K.D., "A soluble polymer-bound approach to the Sharpless catalytic asymmetric dihydroxylation (AD) reaction: Preparation and application of a [(DHQD)2 PHAL-PEG-OMe] ligand"
Tetrahedron Letters, 38, 1527 (1997) |
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Zhao, X.-Y., Jung, K.W., Janda, K.D., "Soluble polymer synthesis: An improved traceless linker methodology for aliphatic C-H bond formation"
Tetrahedron Letters, 38, 977 (1997) |
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